SCHEMBL17090197

SCHEMBL17090197

Cc1c(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)C)CC2)ccc(OCC2CC2)c1C

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 2/20 0.36
GRIA2 P42262 5/20 0.36
BRD4 O60885 5/20 0.35
DRD2 P14416 2/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
NPY5R Q15761 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565174 1.00 PTGER4 (0.36) PTGER4GRIA2BRD4DRD2ADRA1D
SCHEMBL13565307 0.88 PTGER4 (0.35) PTGER4GRIA2BRD4MKNK1MKNK2
SCHEMBL17090190 0.88 PTGER4 (0.35) PTGER4GRIA2BRD4MKNK1MKNK2
SCHEMBL17090189 0.85 PDE4A (0.37) PTGER4BRD4PDE4APDE4BPDE4C
SCHEMBL13565127 0.85 PDE4A (0.37) PTGER4BRD4PDE4APDE4BPDE4C
SCHEMBL13204432 0.83 GSK3A (0.38) GRIA2PDE4APDE4BPDE4CPDE4D
SCHEMBL10114950 0.83 GSK3A (0.38) GRIA2PDE4APDE4BPDE4CPDE4D
SCHEMBL13564939 0.82 ACACB (0.39) PTGER4GRIA2BRD4NPY5R
SCHEMBL17090034 0.82 ACACB (0.39) PTGER4GRIA2BRD4NPY5R
SCHEMBL11941027 0.80 GRIA2 (0.38) GRIA2BRD4DRD2ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed