SCHEMBL17090263

SCHEMBL17090263

CCC(C)(C)S(=O)(=O)N[C@H]1CC[C@H](CNc2ccc(N3C[C@@H](C)O[C@@H](C)C3)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.40
LRRK2 Q5S007 9/20 0.39
CNR2 P34972 3/20 0.34
HTR2A P28223 2/20 0.34
DRD3 P35462 2/20 0.34
BTK Q06187 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALDH3A1 P30838 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565844 1.00 MAPT (0.40) MAPTLRRK2CNR2HTR2ADRD3
SCHEMBL13565789 0.92 LRRK2 (0.40) MAPTLRRK2CNR2HTR2ADRD3
SCHEMBL17090254 0.92 LRRK2 (0.40) MAPTLRRK2CNR2HTR2ADRD3
SCHEMBL13564738 0.92 MAPT (0.43) MAPTLRRK2CNR2HTR2ADRD3
SCHEMBL13565140 0.92 MAPT (0.43) MAPTLRRK2CNR2HTR2ADRD3
SCHEMBL17089987 0.92 MAPT (0.43) MAPTLRRK2CNR2HTR2ADRD3
SCHEMBL11936149 0.92 MAPT (0.43) MAPTLRRK2CNR2HTR2ADRD3
SCHEMBL11936184 0.86 MAPT (0.43) MAPTLRRK2HTR2ADRD3
SCHEMBL13565767 0.85 ALDH1A1 (0.39) MAPTCNR2ALDH1A1ALDH3A1
SCHEMBL17090219 0.85 MAPT (0.44) MAPTLRRK2HTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed