SCHEMBL17090481

SCHEMBL17090481

CC(C)(C)S(=O)(=O)N[C@H]1CC[C@H](CNc2cccnc2Oc2ccc(F)cc2F)CC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
HTR1A P08908 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CARM1 Q86X55 2/20 0.42
P2RY1 P47900 7/20 0.41
PRMT6 Q96LA8 1/20 0.41
CRHR1 P34998 1/20 0.38
BRD4 O60885 1/20 0.38
CNR2 P34972 2/20 0.37
CNR1 P21554 1/20 0.37
GPR6 P46095 1/20 0.37
TRPA1 O75762 1/20 0.36
ROCK2 O75116 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565603 1.00 MAPT (0.46) MAPTHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL13565874 0.88 MAPT (0.46) MAPTHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL13203773 0.83 MAPT (0.54) MAPTHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL10133358 0.83 MAPT (0.54) MAPTHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL13438694 0.82 MAPT (0.50) MAPTHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL11934828 0.82 MAPT (0.50) MAPTHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL13438991 0.80 CNR2 (0.49) SLC6A3CNR2CNR1
SCHEMBL11935299 0.80 CNR2 (0.49) SLC6A3CNR2CNR1
SCHEMBL13565656 0.77 MAPT (0.49) MAPTHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL11935231 0.76 CNR2 (0.43) CRHR1CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed