SCHEMBL17090546

SCHEMBL17090546

C[C@@H]1CN(c2cc(F)ccc2NCCCCCNS(=O)(=O)C(C)(C)C)C[C@H](C)O1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.35
ALDH1A1 P00352 2/20 0.33
WDR5 P61964 2/20 0.33
NR3C1 P04150 2/20 0.33
NR3C2 P08235 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 3/20 0.32
HTT P42858 2/20 0.32
LMNA P02545 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
MEN1 O00255 1/20 0.32
PKM P14618 1/20 0.32
KMT2A Q03164 1/20 0.32
PIK3CA P42336 1/20 0.32
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
BRD4 O60885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565988 1.00 NPY5R (0.35) NPY5RALDH1A1WDR5NR3C1NR3C2
SCHEMBL13564951 0.86 NPY5R (0.42) NPY5RALDH1A1WDR5TRPV1BRD4
SCHEMBL17090541 0.86 NPY5R (0.42) NPY5RALDH1A1WDR5TRPV1BRD4
SCHEMBL10133498 0.86 HDAC3 (0.46) ALDH1A1WDR5MEN1KMT2A
SCHEMBL10115040 0.86 HDAC3 (0.46) ALDH1A1WDR5MEN1KMT2A
SCHEMBL17090442 0.85 NPY5R (0.34) NPY5RKDM4EHTTLMNATRPV1
SCHEMBL13565327 0.85 NPY5R (0.34) NPY5RKDM4EHTTLMNATRPV1
SCHEMBL17090204 0.84 BRD4 (0.38) NPY5RTRPV1POLBMAPTBRD4
SCHEMBL11935630 0.84 NPY5R (0.35) NPY5RALDH1A1KDM4ELMNAMAPT
SCHEMBL11941032 0.84 NPY5R (0.35) NPY5RALDH1A1KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed