SCHEMBL17090557

SCHEMBL17090557

C[C@H]1CN(c2ccc(NCc3ccc(NS(=O)(=O)C(C)(C)C)cc3)cc2)C(F)[C@@H](C)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.34
L3MBTL1 Q9Y468 5/20 0.34
RAB9A P51151 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
NPC1 O15118 1/20 0.34
KDM4E B2RXH2 5/20 0.33
MAPT P10636 5/20 0.33
ALOX15 P16050 5/20 0.33
ALOX12 P18054 5/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
GFER P55789 2/20 0.33
ALDH1A1 P00352 5/20 0.32
MAPK1 P28482 3/20 0.32
TDP1 Q9NUW8 3/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
KMT2A Q03164 3/20 0.31
ADRB3 P13945 2/20 0.31
MEN1 O00255 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13566052 1.00 GAA (0.34) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL13565301 0.90 GAA (0.35) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL11936120 0.86 GAA (0.36) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL11941038 0.86 GAA (0.36) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL17090480 0.83 MAPT (0.44) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL13105770 0.83 MAPT (0.44) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL17090550 0.83 MAPT (0.44) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL13564992 0.83 MAPT (0.44) GAAL3MBTL1RAB9ACA1CA2
SCHEMBL11935995 0.82 GAA (0.39) GAAL3MBTL1RAB9ANPC1KDM4E
SCHEMBL11941037 0.82 GAA (0.39) GAAL3MBTL1RAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed