SCHEMBL17100110

SCHEMBL17100110

NC(=O)C1(C(N)=O)CCCCOC1=O

nearest known ligand 0.42

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL822058 0.82 CA1 (0.33) CA1CA9
SCHEMBL28549225 0.78 ALDH1A1 (0.31) CA1CA9
SCHEMBL16039711 0.71 KDM4E (0.33) CA1CA9
SCHEMBL35964 0.70 CA1 (0.37) CA1CA9
SCHEMBL4950591 0.70 CA1 (0.37) CA1CA9
Bicarbonate SCHEMBL16553371 0.69 CA1 (0.33) CA1CA9
SCHEMBL7112607 0.69 CA1 (0.40) CA1CA9
SCHEMBL715504 0.68 CA1 (0.36) CA1CA9
SCHEMBL1747628 0.67 CA1 (0.39) CA1CA9
SCHEMBL430902 0.67 CA1 (0.39) CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230013441-A1 METHOD FOR MANUFACTURING A POLYESTER CONTAINING AT LEAST ONE 1,4:3,6-DIANHYDROHEXITOL UNIT WITH REDUCED COLOURING AND IMPROVED RATES OF INCORPORATION OF THE UNIT(S) ROQUETTE FRERES (FR) 2023-01-19 US disclosed
EP-3212692-B1 METHOD FOR PRODUCING A POLYESTER CONTAINING AT LEAST ONE 1,4:3,6-DIANHYDROHEXITOL UNIT WITH IMPROVED COLOURING ROQUETTE FRERES (FR) 2022-04-27 EP disclosed
WO-2021123655-A1 METHOD FOR MANUFACTURING A POLYESTER CONTAINING AT LEAST ONE 1,4:3,6-DIANHYDROHEXITOL UNIT WITH REDUCED COLOURING AND IMPROVED RATES OF INCORPORATION OF THE UNIT(S) ROQUETTE FRERES (FR) 2021-06-24 WO disclosed
CN-107148438-B Process for producing polyesters containing at least one 1,4:3, 6-dianhydrohexitol unit with improved coloration 罗盖特公司 2020-02-28 CN disclosed
EP-3119831-B1 POLYESTERS COMPRISING 2,5-FURANDICARBOXYLATE AND SATURATED DIOL UNITS HAVING A HIGH GLASS TRANSITION TEMPERATURE FURANIX TECHNOLOGIES BV (NL) 2019-10-02 EP disclosed
US-10400062-B2 Method for producing a polyester containing at least one 1,4:3,6-dianhydrohexitol unit with improved colouring ROQUETTE FRERES (FR) 2019-09-03 US disclosed
US-10316140-B2 Polyesters comprising 2,5-furandicarboxylate and saturated diol units having a high glass transition temperature FURANIX TECHNOLOGIES B.V. (NL) 2019-06-11 US disclosed
EP-3143068-B1 THERMOPLASTIC AROMATIC POLYESTERS COMPRISING TETRAHYDROFURAN-DIMETHANOL AND FURANDICARBOXYLIC ACID MOTIFS ROQUETTE FRERES (FR) 2018-05-02 EP disclosed
US-20170335055-A1 METHOD FOR PRODUCING A POLYESTER CONTAINING AT LEAST ONE 1,4:3,6-DIANHYDROHEXITOL UNIT WITH IMPROVED COLOURING ROQUETTE FRERES (FR) 2017-11-23 US disclosed
EP-3212692-A1 METHOD FOR PRODUCING A POLYESTER CONTAINING AT LEAST ONE 1,4:3,6-DIANHYDROHEXITOL UNIT WITH IMPROVED COLOURING Roquette Frères (FR) 2017-09-06 EP disclosed
US-20170190832-A1 THERMOPLASTIC AROMATIC POLYESTERS COMPRISING TETRAHYDROFURAN-DIMETHANOL MOTIFS ROQUETTE FRERES (FR) 2017-07-06 US disclosed
US-20170145153-A1 THERMOPLASTIC AROMATIC POLYESTERS COMPRISING TETRAHYDROFURAN-DIMETHANOL AND FURANDICARBOXYLIC ACID MOTIFS ROQUETTE FRERES (FR) 2017-05-25 US disclosed
US-20170129994-A1 POLYESTERS COMPRISING 2,5-FURANDICARBOXYLATE AND SATURATED DIOL UNITS HAVING A HIGH GLASS TRANSITION TEMPERATURE FURANIX TECHNOLOGIES B.V. (NL) 2017-05-11 US disclosed
EP-3143068-A1 THERMOPLASTIC AROMATIC POLYESTERS COMPRISING TETRAHYDROFURAN-DIMETHANOL AND FURANDICARBOXYLIC ACID MOTIFS Roquette Frères (FR) 2017-03-22 EP disclosed
EP-3140339-A1 THERMOPLASTIC AROMATIC POLYESTERS COMPRISING TETRAHYDROFURAN-DIMETHANOL MOTIFS Roquette Frères (FR) 2017-03-15 EP disclosed
EP-3119831-A1 POLYESTERS COMPRISING 2,5-FURANDICARBOXYLATE AND SATURATED DIOL UNITS HAVING A HIGH GLASS TRANSITION TEMPERATURE Furanix Technologies B.V. (NL) 2017-01-25 EP disclosed
WO-2016066956-A1 METHOD FOR PRODUCING A POLYESTER CONTAINING AT LEAST ONE 1,4:3,6-DIANHYDROHEXITOL UNIT WITH IMPROVED COLOURING ROQUETTE FRERES (FR) 2016-05-06 WO disclosed
WO-2015170050-A1 THERMOPLASTIC AROMATIC POLYESTERS COMPRISING TETRAHYDROFURAN-DIMETHANOL AND FURANDICARBOXYLIC ACID MOTIFS ROQUETTE FRERES (FR) 2015-11-12 WO disclosed
WO-2015170049-A1 THERMOPLASTIC AROMATIC POLYESTERS COMPRISING TETRAHYDROFURAN-DIMETHANOL MOTIFS ROQUETTE FRERES (FR) 2015-11-12 WO disclosed
WO-2015142181-A1 POLYESTERS COMPRISING 2,5-FURANDICARBOXYLATE AND SATURATED DIOL UNITS HAVING A HIGH GLASS TRANSITION TEMPERATURE FURANIX TECHNOLOGIES B.V. (NL) 2015-09-24 WO disclosed