SCHEMBL1710200

SCHEMBL1710200

COc1cc(Cl)c(COC2CCCCO2)c(Cl)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
KDM4C Q9H3R0 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
P2RX3 P56373 6/20 0.33
ICAM1 P05362 1/20 0.32
SELE P16581 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1710212 0.91 NPC1 (0.36) NPC1RAB9AKDM4CL3MBTL1PDE4A
SCHEMBL1710353 0.87 NPC1 (0.39) NPC1RAB9AKDM4CL3MBTL1PDE4A
SCHEMBL1710278 0.85 NPC1 (0.38) NPC1RAB9AKDM4CL3MBTL1PDE4A
SCHEMBL1710252 0.85 KDM4C (0.39) NPC1RAB9AKDM4CL3MBTL1CCNA2
SCHEMBL1710294 0.85 KDM4C (0.40) NPC1RAB9AKDM4CL3MBTL1CCNA2
SCHEMBL1710209 0.77 KDM4C (0.33) NPC1RAB9AKDM4CL3MBTL1P2RX3
SCHEMBL1710182 0.76 NPC1 (0.38) NPC1RAB9AKDM4CL3MBTL1PDE4A
SCHEMBL1563782 0.76 PDE4D (0.41) NPC1RAB9AKDM4CL3MBTL1PDE4A
SCHEMBL1563149 0.74 KDM4C (0.40) NPC1RAB9AKDM4CL3MBTL1PDE4A
SCHEMBL1564674 0.74 PDE4D (0.41) NPC1RAB9AKDM4CL3MBTL1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344477-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS Jerini AG (DE) 2011-07-20 EP disclosed
WO-2010031589-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-03-25 WO disclosed