SCHEMBL1710342

SCHEMBL1710342

C=Cc1nc(C)cc(Cl)c1COC1CCCCO1.Cc1cc(Cl)c(COC2CCCCO2)c(CO)n1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KDM4C Q9H3R0 1/20 0.31
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1562973 0.92 KDM4C (0.35) NPC1RAB9AKDM4C
SCHEMBL1710182 0.91 NPC1 (0.38) NPC1RAB9AKDM4C
SCHEMBL1710209 0.88 KDM4C (0.33) NPC1RAB9AKDM4C
SCHEMBL1710278 0.82 NPC1 (0.38) NPC1RAB9AKDM4CPTPN1
SCHEMBL1710353 0.79 NPC1 (0.39) NPC1RAB9AKDM4C
SCHEMBL1710212 0.78 NPC1 (0.36) NPC1RAB9AKDM4CPTPN1
SCHEMBL1710180 0.78 NPC1 (0.40) NPC1RAB9AKDM4CPTPN1
SCHEMBL1710252 0.78 KDM4C (0.39) NPC1RAB9AKDM4C
SCHEMBL3125092 0.74 NPC1 (0.36) NPC1RAB9AKDM4CPTPN1
SCHEMBL2937355 0.73 NPC1 (0.34) NPC1RAB9AKDM4CPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344477-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS Jerini AG (DE) 2011-07-20 EP disclosed
WO-2010031589-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-03-25 WO disclosed