SCHEMBL17110978

SCHEMBL17110978

C#CC(CC)(NC(=O)c1cc(F)cnc1NC1CCC(F)(F)CC1)S(C)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.43
IRAK4 Q9NWZ3 9/20 0.36
SCN9A Q15858 4/20 0.34
ANO1 Q5XXA6 1/20 0.34
MAPK8 P45983 1/20 0.33
SCN5A Q14524 1/20 0.33
HSD11B1 P28845 1/20 0.32
MAPK1 P28482 1/20 0.31
TDO2 P48775 1/20 0.31
KDM1A O60341 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17110976 1.00 TRPA1 (0.43) TRPA1IRAK4SCN9AANO1MAPK8
SCHEMBL17110910 0.85 TRPA1 (0.46) TRPA1IRAK4SCN9AANO1MAPK8
SCHEMBL17112615 0.85 TRPA1 (0.46) TRPA1IRAK4SCN9AANO1MAPK8
SCHEMBL17110903 0.85 TRPA1 (0.46) TRPA1IRAK4SCN9AANO1MAPK8
SCHEMBL17110894 0.80 TRPA1 (0.49) TRPA1IRAK4ANO1MAPK8
SCHEMBL17110897 0.80 TRPA1 (0.49) TRPA1IRAK4ANO1MAPK8
SCHEMBL17110984 0.80 TRPA1 (0.49) TRPA1IRAK4ANO1MAPK8
SCHEMBL17110980 0.78 TRPA1 (0.45) TRPA1IRAK4ANO1MAPK8MAPK1
SCHEMBL15639912 0.77 TRPA1 (0.71) TRPA1IRAK4
SCHEMBL15638540 0.76 TRPA1 (0.56) TRPA1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015144977-A1 TRPA1 MODULATORS ORIEN CORPORATION (FI) 2015-10-01 WO disclosed