SCHEMBL17112012

SCHEMBL17112012

O=C(O)c1ccc(C(F)(F)F)c(-c2ccnn2C2CCCCO2)c1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.48
CYP4A11 Q02928 3/20 0.48
ATR Q13535 16/20 0.44
PIK3CD O00329 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17110684 0.89 CYP4F2 (0.45) CYP4F2CYP4A11ATR
SCHEMBL17110705 0.79 NTRK1 (0.59)
SCHEMBL17110606 0.76 ATR (0.45) CYP4F2CYP4A11ATR
SCHEMBL19881080 0.76 CYP4F2 (0.48) CYP4F2CYP4A11ATR
SCHEMBL17110607 0.76 CYP4F2 (0.46) CYP4F2CYP4A11ATR
SCHEMBL17110659 0.75 CYP4F2 (0.43) CYP4F2CYP4A11ATR
SCHEMBL15016182 0.74 CYP4F2 (0.50) CYP4F2CYP4A11ATR
SCHEMBL25261997 0.74 CYP4F2 (0.44) CYP4F2CYP4A11ATR
SCHEMBL15388562 0.73 CYP4F2 (0.46) CYP4F2CYP4A11ATR
SCHEMBL15388563 0.73 CYP4F2 (0.46) CYP4F2CYP4A11ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3122343-A2 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF Merck Sharp & Dohme Corp. (US) 2017-02-01 EP disclosed
EP-3122344-A2 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF Merck Sharp & Dohme Corp. (US) 2017-02-01 EP disclosed
WO-2015148354-A2 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME CORP. (US) 2015-10-01 WO disclosed
WO-2015148350-A2 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME CORP. (US) 2015-10-01 WO disclosed