SCHEMBL17115508

SCHEMBL17115508

CC1(C)CC(c2ccncc2N)C[C@H](N2C(=O)c3ccccc3C2=O)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.34
ALDH1A1 P00352 3/20 0.34
PIM1 P11309 5/20 0.33
PIM3 Q86V86 5/20 0.33
PIM2 Q9P1W9 5/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
TMEM97 Q5BJF2 2/20 0.32
HTR2A P28223 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
HTR2B P41595 1/20 0.32
ALOX15 P16050 1/20 0.32
HTT P42858 1/20 0.32
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
NOS2 P35228 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2692672 1.00 TSHR (0.34) TSHRALDH1A1PIM1PIM3PIM2
SCHEMBL2694105 1.00 TSHR (0.34) TSHRALDH1A1PIM1PIM3PIM2
SCHEMBL2694107 1.00 TSHR (0.34) TSHRALDH1A1PIM1PIM3PIM2
SCHEMBL2692676 1.00 TSHR (0.34) TSHRALDH1A1PIM1PIM3PIM2
SCHEMBL1723165 1.00 TSHR (0.34) TSHRALDH1A1PIM1PIM3PIM2
SCHEMBL15338281 0.81
SCHEMBL1723397 0.81 ALDH1A1 (0.40) ALDH1A1PIM1PIM3PIM2ADRA1D
SCHEMBL13833169 0.81 ALDH1A1 (0.40) ALDH1A1PIM1PIM3PIM2ADRA1D
SCHEMBL13833170 0.81 ALDH1A1 (0.40) ALDH1A1PIM1PIM3PIM2ADRA1D
SCHEMBL2694268 0.74 PIM1 (0.45) ALDH1A1PIM1PIM3PIM2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344474-B1 PICOLINAMIDE DERIVATIVES AS KINASE INHIBITORS NOVARTIS AG (CH) 2015-09-23 EP disclosed