SCHEMBL1711961

SCHEMBL1711961

CCOC(=O)N1C[C@H]2CNCC1C2

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNA4 P43681 19/20 0.47
CHRNB2 P17787 18/20 0.47
CHRNB4 P30926 16/20 0.47
CHRNA3 P32297 16/20 0.47
CHRNA7 P36544 13/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1711611 1.00 CHRNA4 (0.47) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL1710945 1.00 CHRNA4 (0.47) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL2546530 1.00 CHRNA4 (0.47) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL2958380 0.87 CHRNB2 (0.41) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL2653632 0.84 KMT2A (0.40) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL1711273 0.83 CHRNB2 (0.64) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL2540484 0.83 CHRNB2 (0.64) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL1711197 0.83 CHRNB2 (0.64) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL2546533 0.79 CHRNB2 (0.64) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL17039078 0.79 GAA (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344496-A1 AMIDES OF DIAZABICYCLOOCTANES AND USES THEREOF Targacept Inc. (US) 2011-07-20 EP disclosed
WO-2010028033-A1 AMIDES OF DIAZABICYCLOOCTANES AND USES THEREOF TARGACEPT, INC. (US) 2010-03-11 WO disclosed