SCHEMBL171226

SCHEMBL171226

N#Cc1cccc(Cc2ccncc2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.56
CYP11B1 P15538 5/20 0.53
CYP11B2 P19099 5/20 0.53
CYP19A1 P11511 4/20 0.53
GSK3A P49840 1/20 0.50
GSK3B P49841 1/20 0.50
LRRK2 Q5S007 1/20 0.46
GLA P06280 1/20 0.44
MPO P05164 1/20 0.44
NAMPT P43490 1/20 0.44
IDH1 O75874 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
CYP17A1 P05093 3/20 0.42
CYP3A4 P08684 3/20 0.42
AKT1 P31749 1/20 0.42
LTA4H P09960 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2153847 0.87 HRH3 (0.59) HRH3CYP11B1CYP11B2CYP19A1GSK3B
SCHEMBL4196662 0.85 HRH3 (0.54) HRH3CYP11B1CYP11B2CYP19A1GLA
SCHEMBL171388 0.83 HRH3 (0.57) HRH3CYP11B1CYP11B2CYP19A1NAMPT
SCHEMBL29442890 0.83 HRH3 (0.57) HRH3CYP11B1CYP11B2CYP19A1NAMPT
SCHEMBL171234 0.79 HRH3 (0.53) HRH3CYP11B1CYP11B2CYP19A1GSK3A
SCHEMBL481239 0.79 HRH3 (0.49) HRH3CYP11B1CYP11B2CYP19A1GLA
SCHEMBL26987873 0.79 HRH3 (0.49) HRH3CYP11B1CYP11B2CYP19A1GSK3B
SCHEMBL18641329 0.76 HRH3 (0.50) HRH3CYP11B1CYP11B2CYP19A1GLA
SCHEMBL18641315 0.75 LTA4H (0.58) HRH3GLAIDH1CLK4LTA4H
SCHEMBL28085045 0.75 HRH3 (0.49) HRH3CYP11B1CYP11B2CYP19A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426122-A1 Methylene urea derivative as RAF kinasse inhibitors Merck Patent GmbH (DE) 2012-03-07 EP disclosed