SCHEMBL1713091

SCHEMBL1713091

C#Cc1c(C(=O)O)ccc(C(=O)O)c1-c1cccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.54
PTPN22 Q9Y2R2 1/20 0.54
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 1/20 0.49
HPGD P15428 1/20 0.49
NR4A1 P22736 1/20 0.49
NR4A2 P43354 1/20 0.49
NR4A3 Q92570 1/20 0.49
MCL1 Q07820 2/20 0.47
ACMSD Q8TDX5 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LDHA P00338 1/20 0.45
CDC25B P30305 1/20 0.44
SOS1 Q07889 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HSD17B10 Q99714 1/20 0.40
RORC P51449 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1713092 0.85 PTPN22 (0.56) WDR5PTPN22ALDH1A1KDM4EHPGD
SCHEMBL1712748 0.84 PTPN22 (0.53) WDR5PTPN22ALDH1A1KDM4EHPGD
SCHEMBL9124028 0.82 WDR5 (0.79) WDR5ALDH1A1KDM4EHPGDNR4A1
SCHEMBL29458346 0.82 WDR5 (0.79) WDR5ALDH1A1KDM4EHPGDNR4A1
SCHEMBL1713101 0.77 PTPN22 (0.52) WDR5PTPN22ALDH1A1KDM4EHPGD
SCHEMBL21638943 0.76 PTPN22 (0.46) WDR5PTPN22ALDH1A1KDM4EMCL1
SCHEMBL9750103 0.76 MCL1 (0.60) WDR5PTPN22ALDH1A1KDM4EHPGD
SCHEMBL29795098 0.74 WDR5 (0.74) WDR5ALDH1A1KDM4EHPGDNR4A1
SCHEMBL28044056 0.74 MYC (0.65) WDR5ALDH1A1KDM4EHPGDNR4A1
SCHEMBL2651037 0.73 MCL1 (0.57) WDR5PTPN22ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344568-B1 ACETYLENIC POLYAMIDE NEXAM CHEMICAL AB (SE) 2017-12-20 EP claimed
US-8492507-B2 Acetylenic polyamide NEXAM CHEMICAL AB (SE) 2013-07-23 US claimed
US-20110190469-A1 ACETYLENIC POLYAMIDE NEXAM CHEMICAL AB (SE) 2011-08-04 US claimed
EP-2344568-A1 ACETYLENIC POLYAMIDE Nexam Chemical AB (SE) 2011-07-20 EP claimed
WO-2010036170-A1 ACETYLENIC POLYAMIDE NEXAM CHEMICAL AB (SE) 2010-04-01 WO claimed
WO-2010030216-A1 ACETYLENIC POLY(ALKYLENE PHTHALATE) NEXAM CHEMICAL AB (SE) 2010-03-18 WO claimed
EP-3907247-B1 GLASS TRANSITION HIGH-TEMPERATURE SEMI-CRYSTALLINE POLYAMIDE COMPOSITION MADE OF NEAR-FIELD DIAMINE FOR THERMOPLASTIC MATERIAL, METHOD FOR MANUFACTURING SAME AND USES THEREOF ARKEMA FRANCE (FR) 2023-08-16 EP disclosed
EP-4159792-A1 SEMI-CRYSTALLINE POLYAMIDE COMPOSITION WITH A HIGH GLASS TRANSITION TEMPERATURE BASED ON SHORT DIAMINE FOR THERMOPLASTIC MATERIAL, METHOD FOR MAKING SAME AND USES THEREOF ARKEMA FRANCE (FR) 2023-04-05 EP disclosed
EP-3601410-A1 SHORT DIAMINE-BASED SEMI-CRYSTALLINE POLYAMIDE COMPOSITION HAVING A HIGH GLASS TRANSITION TEMPERATURE FOR A THERMOPLASTIC MATERIAL, PRODUCTION METHOD THEREOF AND USES OF SAME Arkema France (FR) 2020-02-05 EP disclosed
EP-3443022-A1 SEMI-CRYSTALLINE POLYAMIDE COMPOSITION HAVING A HIGH GLASS TRANSITION TEMPERATURE AND A HIGH MELTING TEMPERATURE FOR A THERMOPLASTIC MATERIAL, PRODUCTION METHOD THEREOF AND USES OF SAME Arkema France (FR) 2019-02-20 EP disclosed
EP-3325537-A1 SEMI-CRYSTALLINE POLYAMIDE COMPOSITION HAVING A HIGH GLASS TRANSITION TEMPERATURE FOR A THERMOPLASTIC MATERIAL, PRODUCTION METHOD THEREOF AND USES OF SAME Arkema France (FR) 2018-05-30 EP disclosed
EP-3325538-A1 SEMI-CRYSTALLINE POLYAMIDE COMPOSITION HAVING A HIGH GLASS TRANSITION TEMPERATURE FOR A COMPOSITE MATERIAL, PRODUCTION METHOD THEREOF AND USES OF SAME Arkema France (FR) 2018-05-30 EP disclosed
EP-2344568-B1 ACETYLENIC POLYAMIDE NEXAM CHEMICAL AB (SE) 2017-12-20 EP disclosed
US-8492507-B2 Acetylenic polyamide NEXAM CHEMICAL AB (SE) 2013-07-23 US disclosed
US-20110190469-A1 ACETYLENIC POLYAMIDE NEXAM CHEMICAL AB (SE) 2011-08-04 US disclosed
EP-2344568-A1 ACETYLENIC POLYAMIDE Nexam Chemical AB (SE) 2011-07-20 EP disclosed
WO-2010036170-A1 ACETYLENIC POLYAMIDE NEXAM CHEMICAL AB (SE) 2010-04-01 WO disclosed
WO-2010030216-A1 ACETYLENIC POLY(ALKYLENE PHTHALATE) NEXAM CHEMICAL AB (SE) 2010-03-18 WO disclosed