SCHEMBL171379

SCHEMBL171379

CCc1nc2c(N)nc(SC(c3ccccc3)c3ccccc3)nc2n1C

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.37
ADORA2A P29274 8/20 0.37
ADORA2B P29275 6/20 0.37
TLR7 Q9NYK1 3/20 0.36
PI4KA P42356 2/20 0.35
PI4K2B Q8TCG2 2/20 0.35
PI4K2A Q9BTU6 2/20 0.35
PI4KB Q9UBF8 2/20 0.35
ADORA3 P0DMS8 3/20 0.33
FYN P06241 1/20 0.33
TMIGD3 P0DMS9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL97827 0.78 PIK3CA (0.51)
SCHEMBL5162427 0.67 ABCB1 (0.48) ADORA1ADORA2AADORA2BTLR7PI4KA
SCHEMBL171439 0.65 SMN1; SMN2 (0.35)
SCHEMBL5177679 0.65 PI4KA (0.46) ADORA1ADORA2AADORA2BTLR7PI4KA
SCHEMBL25093187 0.64 TLR7 (0.67) TLR7
SCHEMBL3441083 0.64 RXFP1 (0.45) ADORA1ADORA2AADORA2BTLR7
SCHEMBL17442995 0.62 HSP90AA1 (0.45) ADORA1ADORA2AADORA2BTLR7PI4KA
SCHEMBL3441050 0.62 PI4KA (0.49) ADORA1ADORA2AADORA2BTLR7PI4KA
SCHEMBL5160564 0.62 ABCB1 (0.51) ADORA1ADORA2AADORA2BADORA3TMIGD3
SCHEMBL449339 0.61 AKT1 (0.38) ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed