SCHEMBL171439

SCHEMBL171439

CCOc1ccc(CSc2nc(N)c3nc(CC)n(C)c3n2)cc1N

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.35
ALOX12 P18054 1/20 0.35
ALDH1A1 P00352 5/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
MAPT P10636 3/20 0.34
LMNA P02545 3/20 0.34
NPC1 O15118 3/20 0.34
TSHR P16473 3/20 0.34
USP2 O75604 2/20 0.34
RECQL P46063 1/20 0.34
HPGD P15428 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
RAB9A P51151 3/20 0.33
HSD17B10 Q99714 1/20 0.33
CREBBP Q92793 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99069 0.84 PIK3CA (0.50) ALDH1A1L3MBTL1LMNAHPGDHSD17B10
SCHEMBL98783 0.79 ALDH1A1 (0.39) SMN1; SMN2ALOX12ALDH1A1L3MBTL1MAPT
SCHEMBL98984 0.77 PIK3CA (0.49) SMN1; SMN2ALDH1A1L3MBTL1LMNAHPGD
SCHEMBL171639 0.76 PAK4 (0.36) ALDH1A1L3MBTL1MAPTLMNA
SCHEMBL98098 0.75 PIK3CA (0.49) ALDH1A1L3MBTL1LMNA
SCHEMBL96510 0.74 YTHDC1 (0.40) ALDH1A1MAPTUSP2HPGD
SCHEMBL99695 0.74 MAPT (0.35) SMN1; SMN2ALDH1A1L3MBTL1MAPTLMNA
SCHEMBL97311 0.74 PDE10A (0.42) ALDH1A1L3MBTL1LMNATSHRHPGD
SCHEMBL97830 0.73 ALDH1A1 (0.34) SMN1; SMN2ALOX12ALDH1A1L3MBTL1
SCHEMBL100087 0.72 PIK3CA (0.46) ALDH1A1L3MBTL1MAPTLMNAUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed