SCHEMBL17149495

SCHEMBL17149495

BC(=O)N1CCC(C#N)(Nc2ccc(Br)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA4 P22748 3/20 0.39
CA5A P35218 3/20 0.39
CA7 P43166 3/20 0.39
CA9 Q16790 3/20 0.39
CA13 Q8N1Q1 3/20 0.39
CA14 Q9ULX7 3/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38
ALDH1A1 P00352 3/20 0.38
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
DUSP3 P51452 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17140737 0.80 JAK2 (0.52) ALDH1A1FPR3FPR2JAK2JAK1
SCHEMBL17140624 0.77 SMN1; SMN2 (0.42) CYP1A2SMN1; SMN2GAARAB9ANPC1
SCHEMBL17149444 0.77 CA12 (0.41) SMN1; SMN2CA12CA1CA2CA4
SCHEMBL28173332 0.75 SMN1; SMN2 (0.48) CYP1A2SMN1; SMN2CA12CA1CA2
SCHEMBL20340406 0.75 CYP1A2 (0.71) CYP1A2SMN1; SMN2GAAALDH1A1LMNA
SCHEMBL4465130 0.74 CYP1A2 (0.45) CYP1A2SMN1; SMN2CA12CA1CA2
SCHEMBL16876701 0.71 SMN1; SMN2 (0.63) SMN1; SMN2CA12CA1CA2CA4
SCHEMBL17140740 0.70 SMN1; SMN2 (0.34) CYP1A2SMN1; SMN2CA12CA1CA2
SCHEMBL11046085 0.69 MAPT (0.47) CYP1A2GAARAB9ANPC1ALDH1A1
SCHEMBL222683 0.69 GPR119 (0.49) SMN1; SMN2CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015154023-A1 SUBSTITUTED SPIROCYDIC INHIBITORS OF AUTOTAXIN X-RX DISCOVERY, INC. (US) 2015-10-08 WO disclosed