SCHEMBL171517

SCHEMBL171517

CCc1ccc(C2=CCCN(C(=O)OCc3ccccc3)C2)nc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CYP2C19 P33261 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TMEM97 Q5BJF2 10/20 0.39
SIGMAR1 Q99720 10/20 0.39
ACKR3 P25106 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14544156 0.86 SMN1; SMN2 (0.42) DHFRSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL13490485 0.84 DHFR (0.39) DHFRSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL13490483 0.81 CYP1A2 (0.50) DHFRSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL171466 0.81 MEN1 (0.44) DHFRSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL13490590 0.78 MEN1 (0.44) DHFRSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL32677921 0.78 MEN1 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL169428 0.78 GRM5 (0.50) DHFRSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL13490472 0.78 MEN1 (0.43) DHFRSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL171515 0.77 KDM1A (0.43) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL13490572 0.77 P2RY12 (0.43) SMN1; SMN2NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426120-A1 Pyridyltetrahydropyridines and pyridylpiperidines, and method of manufacturing them Fujifilm Finechemicals Co., Ltd. (JP) 2012-03-07 EP disclosed