SCHEMBL17155201

SCHEMBL17155201

COC(=O)C1(N2CCC(Oc3cccc(N=O)c3F)CC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
CCR5 P51681 2/20 0.34
KMT2A Q03164 1/20 0.34
EPHX2 P34913 1/20 0.34
WNT3A P56704 1/20 0.34
HRH1 P35367 1/20 0.33
KDM1A O60341 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPY1R P25929 1/20 0.33
NPY2R P49146 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18406816 0.86 OPRL1 (0.39) OPRL1OPRM1OPRD1PDE4APDE4B
SCHEMBL18411395 0.83 OPRL1 (0.37) OPRL1OPRM1OPRD1PDE4APDE4B
SCHEMBL18406815 0.82 SCD (0.39) OPRL1OPRM1OPRD1PDE4APDE4B
SCHEMBL18411501 0.73 EPHX2 (0.50) OPRM1OPRD1CCR5EPHX2HRH1
SCHEMBL17155368 0.69 OPRL1 (0.36) OPRL1OPRM1OPRD1CCR5
SCHEMBL17155353 0.69 SLC6A2 (0.48) OPRM1CCR5KMT2A
SCHEMBL17155077 0.67 MAPK1 (0.42) OPRL1OPRM1CCR5KMT2ASMN1; SMN2
SCHEMBL17155018 0.66 KMT2A (0.37) OPRL1OPRM1OPRD1CCR5KMT2A
SCHEMBL23163989 0.66 ACACB (0.48) KMT2AEPHX2
SCHEMBL29731444 0.66 ACACB (0.48) KMT2AEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015150557-A1 MACROCYLIC PYRIDINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2015-10-08 WO disclosed