SCHEMBL17155353

SCHEMBL17155353

COC(=O)C1(N2CCC(Oc3cccc([N+](=O)[O-])c3)CC2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.48
SLC6A4 P31645 2/20 0.48
SLC6A3 Q01959 2/20 0.48
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
PGR P06401 1/20 0.40
CHRM2 P08172 1/20 0.40
ABCB1 P08183 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
ADRA1A P35348 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18411501 0.83 EPHX2 (0.50) SLC6A2SLC6A4SLC6A3OPRM1KCNH2
SCHEMBL17155367 0.81 PKM (0.47) CCR5NPC1RAB9AMAPTMEN1
SCHEMBL17154975 0.79 CCR5 (0.39) CHRNB2CHRNA4CCR5MAPTMEN1
SCHEMBL9014151 0.78 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL374672 0.78 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL18406815 0.77 SCD (0.39) OPRM1CCR5MAPT
SCHEMBL2481721 0.77 SLC6A2 (0.56) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL27078145 0.76 ACACB (0.46) SLC6A2SLC6A4SLC6A3
SCHEMBL19878954 0.76 SLC6A2 (0.71) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL29739455 0.76 SLC6A2 (0.71) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015150557-A1 MACROCYLIC PYRIDINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2015-10-08 WO disclosed