SCHEMBL1716932

SCHEMBL1716932

CCC(CC=Cc1ccccc1)C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 12/20 0.65
GRIK2 Q13002 12/20 0.65
HTR2A P28223 3/20 0.51
GRIK3 Q13003 1/20 0.50
PAM P19021 1/20 0.50
CTSC P53634 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1716930 1.00 GRIK1 (0.65) GRIK1GRIK2HTR2AGRIK3PAM
(Z)-1,2-Diphenylethene SCHEMBL4230847 0.85 CYP1A2 (0.50) GRIK1GRIK2PAM
(Z)-1,2-Diphenylethene SCHEMBL4230850 0.85 CYP1A2 (0.50) GRIK1GRIK2PAM
SCHEMBL3252010 0.83 GRIK1 (0.57) GRIK1GRIK2HTR2AGRIK3
SCHEMBL3252009 0.83 GRIK1 (0.57) GRIK1GRIK2HTR2AGRIK3
SCHEMBL21987028 0.83 GRIK1 (0.65) GRIK1GRIK2HTR2AGRIK3PAM
SCHEMBL21987027 0.83 GRIK1 (0.65) GRIK1GRIK2HTR2AGRIK3PAM
SCHEMBL3020746 0.82 GRIK1 (0.59) GRIK1GRIK2HTR2AGRIK3PAM
SCHEMBL3020748 0.82 GRIK1 (0.59) GRIK1GRIK2HTR2AGRIK3PAM
SCHEMBL7658428 0.82 GRIK1 (0.60) GRIK1GRIK2HTR2AGRIK3PAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3911172-B1 COMBINATION OF SATIETY COMPONENTS WITH ARGININE SYMRISE AG (DE) 2026-04-15 EP claimed
WO-2017156147-A1 IMMUNE BOOSTING DIETARY COMPOUNDS FOR DISEASE CONTROL AND PREVENTION THE BOARD OF REGENTS FOR OKLAHOMA STATE UNIVERSITY OFFICE OF INTELLECTUAL PROPERTY MANAGEMENT TECHNOLOGY DEVELOPMENT CENTER (US) 2017-09-14 WO claimed
EP-1716159-B1 BICYCLIC SILOXANE COMPOSITIONS FOR THE RELEASE OF ACTIVE INGREDIENTS MOMENTIVE PERFORMANCE MAT INC (US) 2011-07-13 EP claimed
EP-1967080-B1 Non-aldehyde cinnamon flavor and delivery systems therefor CADBURY ADAMS USA LLC (US) 2010-06-02 EP claimed
EP-1697386-B1 ACTIVE INGREDIENT-RELEASING CYCLIC SILOXANES GEN ELECTRIC (US) 2007-10-10 EP claimed
EP-0428276-B1 Acaricidal composition TAKASAGO PERFUMERY CO LTD (JP) 1998-09-16 EP claimed
EP-3911172-B1 COMBINATION OF SATIETY COMPONENTS WITH ARGININE SYMRISE AG (DE) 2026-04-15 EP disclosed
EP-3911172-A1 COMBINATION REMEDY Symrise AG (DE) 2021-11-24 EP disclosed
EP-2145042-B2 TEXTILE SCENTING HENKEL AG & CO KGAA (DE) 2021-10-06 EP disclosed
WO-2020147977-A1 COMBINATION REMEDY SYMRISE AG (DE) 2020-07-23 WO disclosed
EP-3474833-A1 CINNAMYL ALCOHOL DERIVATIVE FOR REDUCING APPETITE AND FOR GENERATING THE FEELING OF BEING FULL Symrise AG (DE) 2019-05-01 EP disclosed
EP-2145042-B1 TEXTILE SCENTING HENKEL AG & CO KGAA (DE) 2018-01-17 EP disclosed
WO-2017220168-A1 CINNAMYL ALCOHOL DERIVATIVE FOR REDUCING APPETITE AND FOR GENERATING THE FEELING OF BEING FULL SYMRISE AG (DE) 2017-12-28 WO disclosed
EP-2145042-A1 TEXTILE SCENTING Henkel AG & Co. KGaA (DE) 2010-01-20 EP disclosed
WO-2008135306-A1 TEXTILE SCENTING HENKEL AG & CO. KGAA (DE) 2008-11-13 WO disclosed
EP-1928992-A1 CONSUMER PRODUCTS HAVING VARYING ODORS Henkel AG & Co. KGaA (DE) 2008-06-11 EP disclosed
EP-1922398-A1 CONSUMER PRODUCTS HAVING VARYING ODOR PATTERNS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2008-05-21 EP disclosed
WO-2007028479-A1 CONSUMER PRODUCTS HAVING VARYING ODORS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2007-03-15 WO disclosed
WO-2007028477-A1 CONSUMER PRODUCTS HAVING VARYING ODOR PATTERNS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2007-03-15 WO disclosed