SCHEMBL1717437

SCHEMBL1717437

CC[C@H](NC(=O)c1c(CN2[C@@H]3CC[C@H]2C[C@H](O)C3)n(-c2ccccc2)c(=O)c2ccccc12)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 17/20 0.43
TACR2 P21452 10/20 0.43
OPRM1 P35372 4/20 0.43
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2D6 P10635 1/20 0.41
TACR1 P25103 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
ALDH1A1 P00352 2/20 0.39
TSHR P16473 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1718239 0.86 TACR3 (0.44) TACR3TACR2OPRM1CYP1A2CYP3A4
SCHEMBL1718029 0.86 TACR3 (0.47) TACR3TACR2OPRM1CYP1A2CYP3A4
SCHEMBL1717604 0.84 TACR3 (0.44) TACR3TACR2OPRM1CYP1A2CYP3A4
SCHEMBL1718010 0.84 TACR3 (0.44) TACR3TACR2OPRM1CYP1A2CYP3A4
SCHEMBL1716817 0.84 TACR3 (0.44) TACR3TACR2OPRM1CYP1A2CYP3A4
SCHEMBL1717850 0.83 TACR3 (0.44) TACR3TACR2OPRM1CYP1A2CYP3A4
SCHEMBL2676363 0.83 HTR3E (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL2676365 0.83 HTR3E (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1719365 0.83 HTR3E (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1719367 0.83 HTR3E (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP disclosed