SCHEMBL1717543

SCHEMBL1717543

CC[C@H](NC(=O)c1c(CN2CCN(c3ccccc3F)CC2)n(-c2ccccc2)c(=O)c2ccccc12)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.46
TACR3 P29371 11/20 0.44
TACR2 P21452 5/20 0.44
OPRM1 P35372 4/20 0.44
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPT P10636 1/20 0.39
USP2 O75604 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1717750 0.92 HTR7 (0.43) HTR7TACR3TACR2OPRM1
SCHEMBL1718058 0.89 TACR3 (0.47) HTR7TACR3TACR2OPRM1
SCHEMBL1717610 0.89 HTR7 (0.49) HTR7TACR3KDM4EALDH1A1HSD17B10
SCHEMBL1718018 0.89 TACR3 (0.43) HTR7TACR3TACR2OPRM1KDM4E
SCHEMBL1718231 0.88 TACR3 (0.49) TACR3TACR2OPRM1KDM4EALDH1A1
SCHEMBL1717288 0.88 TACR3 (0.47) HTR7TACR3TACR2OPRM1
SCHEMBL1718782 0.87 TACR3 (0.50) TACR3TACR2OPRM1
SCHEMBL1719079 0.87 TACR3 (0.56) TACR3TACR2OPRM1MEN1KMT2A
SCHEMBL1717859 0.87 TACR3 (0.48) TACR3TACR2OPRM1KDM4EALDH1A1
SCHEMBL1717555 0.87 TACR3 (0.48) TACR3TACR2OPRM1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP claimed
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP disclosed