SCHEMBL1718356

SCHEMBL1718356

COc1ccc(CNC(=O)c2nn3c(C(F)(F)F)cc(-c4ccccc4)nc3c2Cl)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.74
HPGD P15428 3/20 0.74
NPSR1 Q6W5P4 2/20 0.74
CYP1A2 P05177 1/20 0.74
CYP3A4 P08684 1/20 0.74
CYP2C9 P11712 1/20 0.74
CYP2C19 P33261 1/20 0.74
MAPK1 P28482 1/20 0.59
CASP1 P29466 3/20 0.58
CASP7 P55210 3/20 0.58
GAA P10253 1/20 0.58
RXFP1 Q9HBX9 4/20 0.57
MAPT P10636 7/20 0.55
USP2 O75604 2/20 0.54
PTGES O14684 1/20 0.53
POLB P06746 2/20 0.53
MYC P01106 1/20 0.52
MAX P61244 1/20 0.52
KDM4E B2RXH2 3/20 0.51
TSHR P16473 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1717999 0.97 ALDH1A1 (0.77) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1717821 0.96 ALDH1A1 (0.77) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1718192 0.92 ALDH1A1 (0.73) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1718595 0.92 ALDH1A1 (0.72) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1718638 0.91 MAPK1 (0.66) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1718005 0.90 MAPK1 (0.63) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1717917 0.90 RXFP1 (0.72) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1718636 0.89 MAPK1 (0.62) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1719199 0.88 ALDH1A1 (0.71) ALDH1A1HPGDNPSR1CYP1A2CYP3A4
SCHEMBL1718181 0.86 MAPT (0.73) ALDH1A1HPGDNPSR1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed