SCHEMBL1718809

SCHEMBL1718809

O=C(NC1CCCC1)c1cc2nc(-c3ccccc3)cc(-c3ccccc3)n2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 1.00
HTT P42858 4/20 1.00
ALDH1A1 P00352 7/20 0.64
MAPT P10636 6/20 0.61
MAPK1 P28482 2/20 0.61
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
HPGD P15428 7/20 0.61
LMNA P02545 4/20 0.61
NPSR1 Q6W5P4 3/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
TP53 P04637 4/20 0.60
TDP1 Q9NUW8 1/20 0.59
GAA P10253 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
ADRA2A P08913 1/20 0.54
ADRA2B P18089 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4201226 0.99 KDM4E (0.98) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL25430390 0.98 KDM4E (0.96) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL25969033 0.89 KDM4E (0.80) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL4737182 0.88 KDM4E (0.78) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL25970230 0.88 KDM4E (0.78) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL4215699 0.87 KDM4E (0.77) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL25969141 0.87 KDM4E (0.77) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL14366824 0.86 KDM4E (0.76) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL25338396 0.85 KDM4E (0.74) KDM4EHTTALDH1A1MAPTMAPK1
SCHEMBL25335602 0.85 KDM4E (0.74) KDM4EHTTALDH1A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed