SCHEMBL17188570

SCHEMBL17188570

Cc1cccc(OCC#CCN)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.46
GRM5 P41594 3/20 0.43
DRD2 P14416 2/20 0.43
DRD4 P21917 2/20 0.43
ALDH1A1 P00352 1/20 0.42
DRD3 P35462 1/20 0.42
MAOB P27338 2/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
EGLN1 Q9GZT9 1/20 0.40
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14085290 0.84 ACHE (0.47) ACHEGRM5DRD2DRD4DRD3
SCHEMBL12879342 0.82 ACHE (0.48) ACHEGRM5DRD2DRD4ALDH1A1
SCHEMBL10574546 0.79 ACHE (0.42) ACHEGRM5DRD2DRD4DRD3
SCHEMBL17188576 0.78 GRM5 (0.49) ACHEGRM5DRD2DRD4ALDH1A1
SCHEMBL3982634 0.77 TAAR1 (0.50) ALDH1A1MAOB
SCHEMBL3246350 0.77 ACHE (0.56) ACHEDRD2DRD4ALDH1A1DRD3
SCHEMBL4815490 0.77 MAOB (0.52) ACHEDRD2DRD4ALDH1A1DRD3
SCHEMBL756665 0.77 ACHE (0.50) ACHEDRD2DRD4ALDH1A1DRD3
SCHEMBL8195129 0.77 ACHE (0.50) ACHEDRD2DRD4ALDH1A1DRD3
SCHEMBL7408051 0.74 TAAR1 (0.57) ACHEDRD2DRD4DRD3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9161922-B2 Amine oxidase inhibitors CASE WESTERN RESERVE UNIVERSITY (US) 2015-10-20 US disclosed