SCHEMBL17196243

SCHEMBL17196243

NCc1ccc(N)c(CN)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 6/20 0.46
HRH3 Q9Y5N1 1/20 0.42
ABAT P80404 1/20 0.39
ROCK1 Q13464 1/20 0.38
GAA P10253 2/20 0.38
F10 P00742 1/20 0.38
CYP3A4 P08684 1/20 0.38
PNMT P11086 1/20 0.38
ENPP2 Q13822 1/20 0.38
ST14 Q9Y5Y6 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP2A6 P11509 1/20 0.38
AOC1 P19801 1/20 0.37
AOC3 Q16853 1/20 0.37
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28283960 0.88 GAA (0.52) LOXL2HRH3GAAF10CYP3A4
SCHEMBL27813672 0.84 PRSS1 (0.39) LOXL2ABATGAAF10CYP3A4
SCHEMBL10061520 0.84 TAAR1 (0.41) LOXL2GAACYP3A4KDM4EMEN1
SCHEMBL27892650 0.84 LOXL2 (0.41) LOXL2HRH3ABATROCK1GAA
SCHEMBL15699808 0.84 LOXL2 (0.41) LOXL2HRH3ABATROCK1GAA
SCHEMBL2037286 0.84 CSNK2A1 (0.46) LOXL2HRH3ROCK1GAACYP3A4
SCHEMBL27656591 0.84 CYP3A4 (0.39) LOXL2HRH3ABATGAAF10
SCHEMBL27833864 0.84 LOXL2 (0.36) LOXL2HRH3ABATGAAF10
SCHEMBL28875537 0.82 SKP2 (0.44)
SCHEMBL22106784 0.81 LOXL2 (0.38) LOXL2HRH3ABATROCK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161142-A1 QUINOXALINE COMPOUNDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2015-10-22 WO disclosed