SCHEMBL17196430

SCHEMBL17196430

CCc1cc(C(F)F)nn1C

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.32
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12887815 0.84 KCNH2 (0.30) KCNH2
SCHEMBL10129937 0.83 LRRK2 (0.35) LRRK2
SCHEMBL28156988 0.82
SCHEMBL22275230 0.82
SCHEMBL23736428 0.78 LRRK2 (0.33) LRRK2
SCHEMBL13734950 0.72 CYP11B1 (0.30)
SCHEMBL17072614 0.72
SCHEMBL15100969 0.72 BAZ2B (0.37)
SCHEMBL12203385 0.72 ALDH1A1 (0.33)
SCHEMBL22275476 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015158427-A1 HETEROARYL SUBSTITUTED HETEROCYCLYL SULFONES Grünenthal GmbH (DE) 2015-10-22 WO disclosed