SCHEMBL17196870

SCHEMBL17196870

C=CC(=O)Nc1cc(Nc2ncc(Cl)c(OC3CNC3)n2)c(OC)cc1N1CCN(C)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.68
ALK Q9UM73 3/20 0.62
IGF1R P08069 2/20 0.62
KCNH2 Q12809 2/20 0.62
PLK4 O00444 1/20 0.55
GAK O14976 1/20 0.55
NUAK1 O60285 1/20 0.55
JAK2 O60674 1/20 0.55
FLT3 P36888 1/20 0.55
BLK P51451 1/20 0.55
BMX P51813 1/20 0.55
JAK3 P52333 1/20 0.55
CTSC P53634 1/20 0.55
PTK2 Q05397 1/20 0.55
BTK Q06187 1/20 0.55
ITK Q08881 1/20 0.55
ERBB4 Q15303 1/20 0.55
DCLK3 Q9C098 1/20 0.55
NUAK2 Q9H093 1/20 0.55
EML4 Q9HC35 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17196683 0.88 EGFR (0.65) EGFRALKIGF1RKCNH2PLK4
SCHEMBL17196847 0.88 EGFR (0.63) EGFRALKIGF1RKCNH2
SCHEMBL18657398 0.85 EGFR (0.69) EGFRIGF1RKCNH2JAK2JAK3
SCHEMBL18657453 0.85 EGFR (0.69) EGFRIGF1RKCNH2JAK2JAK3
SCHEMBL17467224 0.84 EGFR (0.69) EGFRIGF1RKCNH2JAK3
SCHEMBL18657447 0.83 EGFR (0.55) EGFRALKIGF1RKCNH2
SCHEMBL18359226 0.83 EGFR (0.70) EGFRALKIGF1RKCNH2JAK3
SCHEMBL19027763 0.83 EGFR (0.72) EGFRALKIGF1RKCNH2JAK3
SCHEMBL19027795 0.82 EGFR (0.68) EGFRALKIGF1RKCNH2PLK4
SCHEMBL18369580 0.81 EGFR (0.83) EGFRALKIGF1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015158233-A1 2,3,4,6-TETRA-SUBSTITUTED BENZENE-1,5-DIAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICINAL USE THEREOF 上海海雁医药科技有限公司 2015-10-22 WO disclosed