SCHEMBL18657447

SCHEMBL18657447

C=CC(=O)Nc1cc(Nc2ncc(Cl)c(OC3CN(S(C)(=O)=O)C3)n2)c(OC)cc1N1CCNCC1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.55
ALK Q9UM73 2/20 0.51
IGF1R P08069 2/20 0.50
KCNH2 Q12809 2/20 0.50
INSR P06213 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17196683 0.92 EGFR (0.65) EGFRALKIGF1RKCNH2
SCHEMBL18563173 0.90 EGFR (0.55) EGFRALKIGF1RKCNH2
SCHEMBL17196684 0.90 EGFR (0.66) EGFRIGF1RKCNH2INSR
SCHEMBL18563178 0.89 EGFR (0.61) EGFRIGF1RKCNH2INSR
Formic Acid SCHEMBL18549295 0.88 EGFR (0.64) EGFRIGF1RKCNH2INSR
SCHEMBL17196834 0.86 EGFR (0.66) EGFRIGF1RKCNH2INSR
SCHEMBL17196821 0.86 EGFR (0.66) EGFRIGF1RKCNH2INSR
SCHEMBL18549237 0.86 EGFR (0.66) EGFRIGF1RKCNH2INSR
SCHEMBL18657449 0.85 ALK (0.48) EGFRALK
SCHEMBL17196852 0.85 EGFR (0.67) EGFRIGF1RKCNH2INSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3144292-A1 2,3,4,6-TETRA-SUBSTITUTED BENZENE-1,5-DIAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICINAL USE THEREOF SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD (US) 2017-03-22 EP disclosed