SCHEMBL1720099

SCHEMBL1720099

Nc1nc(N2CCN(C(=O)COc3ccc(Cl)cc3)CC2)c2nc(-c3ccc[n+]([O-])c3)sc2n1.Nc1nc(N2CCN(C(=O)COc3ccc(Cl)cc3)CC2)c2nc(Cc3ccc(Cl)cc3)sc2n1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 7/20 0.67
KCNH2 Q12809 3/20 0.47
CYP3A4 P08684 2/20 0.43
POLB P06746 1/20 0.41
LMNA P02545 3/20 0.38
MAPK1 P28482 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GPR183 P32249 1/20 0.38
ENPP2 Q13822 5/20 0.37
MAPT P10636 2/20 0.37
PKM P14618 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655262 0.94 PI4KB (0.75) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL656634 0.88 PI4KB (0.70) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL654739 0.85 PI4KB (0.83) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL656541 0.84 PI4KB (0.81) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL654589 0.84 PI4KB (0.65) PI4KBKCNH2POLBLMNAMAPK1
SCHEMBL17102776 0.84 PI4KB (0.63) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL653182 0.81 PI4KB (0.82) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL654457 0.81 PI4KB (0.77) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL653167 0.81 PI4KB (0.75) PI4KBKCNH2CYP3A4POLBLMNA
SCHEMBL654471 0.81 PI4KB (0.75) PI4KBKCNH2CYP3A4POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2405973-A2 THIAZOLOPYRIMIDINE MODULATORS AS IMMUNOSUPPRESSIVE AGENTS Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2012-01-18 EP disclosed