SCHEMBL172018

SCHEMBL172018

Cc1nn(-c2ccccc2)cc1CN1CCN(c2nccnc2N2CCC(CN)CC2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.64
DRD4 P21917 5/20 0.64
DRD3 P35462 5/20 0.64
PLA2G7 Q13093 1/20 0.45
MGLL Q99685 1/20 0.45
ABHD6 Q9BV23 1/20 0.45
OPRM1 P35372 3/20 0.45
KCNH2 Q12809 3/20 0.45
OPRK1 P41145 1/20 0.45
CXCR4 P61073 1/20 0.40
KDM4E B2RXH2 5/20 0.40
SYK P43405 1/20 0.39
CTSS P25774 1/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PKM P14618 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12742602 0.90 DRD2 (0.64) DRD2DRD4DRD3PLA2G7MGLL
Hydrochloric Acid SCHEMBL125248 0.89 DRD2 (0.62) DRD2DRD4DRD3PLA2G7MGLL
SCHEMBL12742617 0.88 DRD2 (0.66) DRD2DRD4DRD3PLA2G7MGLL
SCHEMBL12742556 0.87 DRD2 (0.60) DRD2DRD4DRD3PLA2G7MGLL
Hydrochloric Acid SCHEMBL1448869 0.87 DRD2 (0.65) DRD2DRD4DRD3PLA2G7MGLL
Hydrochloric Acid SCHEMBL122848 0.87 DRD2 (0.59) DRD2DRD4DRD3PLA2G7MGLL
SCHEMBL124437 0.82 DRD4 (0.70) DRD2DRD4DRD3PLA2G7MGLL
SCHEMBL172192 0.82 DRD2 (0.58) DRD2DRD4DRD3PLA2G7MGLL
Hydrochloric Acid SCHEMBL121960 0.81 DRD2 (0.57) DRD2DRD4DRD3PLA2G7MGLL
SCHEMBL171928 0.79 DRD2 (0.49) DRD2DRD4DRD3PLA2G7MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2201002-B1 5-HT7 RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2012-03-07 EP disclosed
WO-2009048765-A1 5-HT7 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2009-04-16 WO disclosed