SCHEMBL1720189

SCHEMBL1720189

Cc1nn(-c2ccc(N3CCC(N(C)C)C3)cc2)c2[nH]c(=O)c3ccccc3c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.46
MAPK1 P28482 1/20 0.46
PDGFRB P09619 1/20 0.45
FGFR1 P11362 1/20 0.45
KDR P35968 1/20 0.45
PARP1 P09874 3/20 0.44
KHK P50053 1/20 0.42
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 3/20 0.42
KCNH2 Q12809 1/20 0.42
HTR2B P41595 2/20 0.41
HTR6 P50406 2/20 0.41
ALDH1A1 P00352 2/20 0.40
MCHR1 Q99705 3/20 0.40
HTT P42858 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4070304 0.99 HPGD (0.45) HPGDMAPK1PDGFRBFGFR1KDR
SCHEMBL13901618 0.94 HPGD (0.47) HPGDMAPK1PDGFRBFGFR1KDR
Hydrochloric Acid SCHEMBL1720563 0.93 HPGD (0.46) HPGDMAPK1PDGFRBFGFR1KDR
SCHEMBL10227998 0.82 PARP1 (0.55) HPGDMAPK1PARP1KHKKDM4E
SCHEMBL13901617 0.82 HPGD (0.61) HPGDMAPK1PARP1KHKKDM4E
SCHEMBL10228002 0.81 PARP1 (0.54) HPGDMAPK1PARP1KHKKDM4E
Hydrochloric Acid SCHEMBL1720180 0.81 HPGD (0.60) HPGDMAPK1PARP1KHKKDM4E
Hydrochloric Acid SCHEMBL1719955 0.81 PARP1 (0.54) HPGDMAPK1PARP1KHKKDM4E
Hydrochloric Acid SCHEMBL1720581 0.80 PARP1 (0.53) HPGDMAPK1PARP1KHKKDM4E
SCHEMBL13901616 0.80 HPGD (0.52) HPGDMAPK1PARP1KHKKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1566380-B1 ISOQUINOLINE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI TANABE PHARMA CORP (JP) 2012-01-11 EP disclosed
EP-1566380-B1 ISOQUINOLINE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI TANABE PHARMA CORP (JP) 2012-01-11 EP disclosed
US-7501412-B2 Isoquinoline compounds and medicinal use thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-10 US disclosed
US-7501412-B2 Isoquinoline compounds and medicinal use thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-10 US disclosed