SCHEMBL172052

SCHEMBL172052

Cc1nc2c(o1)CN(C1CC1)CC2

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.38
CD274 Q9NZQ7 2/20 0.38
DPP4 P27487 2/20 0.35
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DRD2 P14416 1/20 0.31
KCNH2 Q12809 1/20 0.31
LMNA P02545 1/20 0.30
BLM P54132 1/20 0.30
PMP22 Q01453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14930366 0.87 DPP4 (0.36) PDCD1CD274DPP4CYP3A4
SCHEMBL8181509 0.72 DPP4 (0.58) PDCD1CD274DPP4KCNH2
SCHEMBL14549685 0.72 DPP4 (0.58) PDCD1CD274DPP4KCNH2
SCHEMBL12706687 0.71 CYP3A4 (0.32) CYP3A4TSHRHSD17B10LMNABLM
SCHEMBL9963385 0.71 ADORA2A (0.38) CYP3A4TSHRHSD17B10LMNABLM
SCHEMBL6369625 0.71 CYP3A4 (0.53) CYP3A4TSHRHSD17B10DRD2KCNH2
SCHEMBL14970359 0.69 NOTUM (0.39) KCNH2
SCHEMBL24585187 0.68 CYP3A4 (0.45) CYP3A4TSHRHSD17B10LMNABLM
SCHEMBL12765092 0.66 DPP4 (0.33) DPP4
SCHEMBL14908332 0.65 ALDH1A1 (0.41) TSHRHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426135-A1 UREA DERIVATIVE HAVING PI3K INHIBITORY ACTIVITY Shionogi&Co., Ltd. (JP) 2012-03-07 EP disclosed