SCHEMBL1720765

SCHEMBL1720765

Nc1nc(N2CCN(C(=O)O)C(Cc3ccccc3)C2)c2nc(-c3ccc(F)cc3)sc2n1.Nc1nc(N2CCN(S(=O)(=O)c3ccccc3)CC2)c2nc(-c3ccc(F)cc3)sc2n1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 4/20 0.42
KCNH2 Q12809 3/20 0.42
CA1 P00915 4/20 0.41
CA2 P00918 4/20 0.41
CA4 P22748 4/20 0.41
CA9 Q16790 4/20 0.41
GBA1 P04062 4/20 0.38
LMNA P02545 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP3A4 P08684 2/20 0.36
PKM P14618 2/20 0.36
GPR6 P46095 1/20 0.36
ALDH1A1 P00352 3/20 0.35
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
GHSR Q92847 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653325 0.92 PI4KB (0.46) PI4KBKCNH2CYP3A4
SCHEMBL653899 0.86 KCNH2 (0.49) PI4KBKCNH2GBA1LMNAALOX15
SCHEMBL1693928 0.77 PI4KB (0.65) PI4KBKCNH2LMNACYP3A4ALDH1A1
SCHEMBL794433 0.74 PI4KB (0.57) PI4KBKCNH2CYP3A4
SCHEMBL655253 0.73 MEN1 (0.51) PI4KBKCNH2LMNACYP3A4ALDH1A1
SCHEMBL653326 0.72 PI4KB (0.56) PI4KBKCNH2LMNAALOX15CYP3A4
SCHEMBL652412 0.70 PI4KB (0.65) PI4KBKCNH2LMNACYP3A4ALDH1A1
SCHEMBL654037 0.69 GBA1 (0.42) PI4KBKCNH2GBA1HPGD
SCHEMBL655068 0.68 PI4KB (0.50) PI4KBKCNH2LMNACYP3A4ALDH1A1
SCHEMBL655537 0.67 PI4KB (0.68) PI4KBKCNH2LMNACYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2405973-A2 THIAZOLOPYRIMIDINE MODULATORS AS IMMUNOSUPPRESSIVE AGENTS Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2012-01-18 EP disclosed