SCHEMBL17209602

SCHEMBL17209602

Cc1ccc(-c2ccc(NC(=O)C3(c4ccc(-c5cnc6[nH]ccc6c5)cc4)CCOCC3)nc2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.45
CD274 Q9NZQ7 1/20 0.44
RIPK1 Q13546 3/20 0.43
MAP4K4 O95819 3/20 0.43
PLK4 O00444 2/20 0.43
ROS1 P08922 2/20 0.43
MARK3 P27448 2/20 0.43
FLT4 P35916 2/20 0.43
KDR P35968 2/20 0.43
CLK2 P49760 2/20 0.43
CSNK1G2 P78368 2/20 0.43
ROCK1 Q13464 2/20 0.43
MINK1 Q8N4C8 2/20 0.43
AURKB Q96GD4 2/20 0.43
PRKD2 Q9BZL6 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
MAP4K5 Q9Y4K4 2/20 0.43
FLT3 P36888 2/20 0.43
JAK2 O60674 1/20 0.43
FGFR1 P11362 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9966373 0.89 CD274 (0.42) CD274RIPK1MAP4K4PLK4ROS1
SCHEMBL9940355 0.87 ABL1 (0.44) CD274RIPK1MAP4K4PLK4ROS1
SCHEMBL14295931 0.86 CD274 (0.42) CD274RIPK1MAP4K4PLK4ROS1
SCHEMBL9966364 0.86 GSK3B (0.49) CD274RIPK1MAP4K4PLK4ROS1
SCHEMBL9966465 0.84 CDK8 (0.43) CD274RIPK1MAP4K4PLK4ROS1
SCHEMBL17210407 0.83 CD274 (0.41) CD274RIPK1MAP4K4PLK4ROS1
SCHEMBL9966527 0.77 PIK3CD (0.48) RIPK1MAP4K4PLK4ROS1MARK3
SCHEMBL9966272 0.76 HDAC1 (0.47) IDO1RIPK1MAP4K4PLK4ROS1
SCHEMBL9966477 0.76 CDK8 (0.46) RIPK1MAP4K4PLK4ROS1MARK3
SCHEMBL9966566 0.74 ABL1 (0.41) MAP4K4HDAC1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651930-B1 BIARYLAMIDE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INT (DE) 2015-10-28 EP disclosed