SCHEMBL1721369

SCHEMBL1721369

CCSc1nc2cc(F)c(F)cc2c(C)c1OC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.34
MAPT P10636 4/20 0.33
THRB P10828 1/20 0.33
KDM4E B2RXH2 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PRNP P04156 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ELANE P08246 4/20 0.33
BCAT2 O15382 1/20 0.33
HSD17B10 Q99714 2/20 0.32
NPC1 O15118 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
RAB9A P51151 1/20 0.32
CASP7 P55210 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
EIF4A1 P60842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1723448 0.88 MAPT (0.35) GAAMAPTKDM4ETDP1ALDH1A1
SCHEMBL1721617 0.81 PTGDR2 (0.38) THRBKDM4ETDP1ALDH1A1RXFP1
SCHEMBL1721367 0.80 PDE10A (0.37) GAAMAPTTHRBKDM4ETDP1
SCHEMBL1722148 0.80 ALDH1A1 (0.35) GAAMAPTTHRBKDM4ETDP1
SCHEMBL3100597 0.77 SMN1; SMN2 (0.40) GAAMAPTKDM4EALDH1A1HSD17B10
SCHEMBL1721273 0.75 TSHR (0.41) GAAMAPTKDM4ETDP1ALDH1A1
SCHEMBL4089333 0.74 KMT2A (0.36) GAAMAPTTHRBKDM4ETDP1
SCHEMBL4088923 0.72 CFTR (0.41) GAAMAPTKDM4ETDP1ALDH1A1
SCHEMBL1723160 0.69 DYRK1A (0.38) MAPTKDM4EALDH1A1ELANEHSD17B10
SCHEMBL1721484 0.69 ELANE (0.41) MAPTELANEHSD17B10NPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406229-A1 SUBSTITUTED 2-MERCAPTOQUINOLINE-3-CARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2012-01-18 EP disclosed
WO-2010102811-A1 SUBSTITUTED 2-MERCAPTOQUINOLINE-3-CARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2010-09-16 WO disclosed