SCHEMBL17224577

SCHEMBL17224577

O=C1NC(C(=O)O)CO1.[LiH]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.39
LMNA P02545 2/20 0.39
BLM P54132 2/20 0.39
ALOX15 P16050 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 1/20 0.39
THRB P10828 1/20 0.39
PMP22 Q01453 1/20 0.39
KMT2A Q03164 1/20 0.39
CAD P27708 2/20 0.36
HTT P42858 1/20 0.36
GRIA2 P42262 1/20 0.35
EGLN1 Q9GZT9 1/20 0.34
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
SLC1A3 P43003 1/20 0.31
SLC1A2 P43004 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1650778 0.98
SCHEMBL6998150 0.98
SCHEMBL756341 0.98
SCHEMBL6186602 0.80
SCHEMBL28763835 0.80
SCHEMBL890128 0.80
SCHEMBL890097 0.80
SCHEMBL1745137 0.78 CYP2D6 (0.36) CYP2D6LMNABLMALOX15CYP1A2
Lithium Ion SCHEMBL17224576 0.78
SCHEMBL1745139 0.78 CYP2D6 (0.36) CYP2D6LMNABLMALOX15CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114031572-A Process for preparing substituted cycloserines 先正达参股股份有限公司 2022-02-11 CN disclosed
US-9815803-B2 Process for the preparation of substituted cycloserines SYNGENTA PARTICIPATIONS AG (CH) 2017-11-14 US disclosed
US-20170204072-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED CYCLOSERINES SYNGENTA PARTICIPATIONS AG (CH) 2017-07-20 US disclosed
US-9643938-B2 Process for the preparation of substituted cycloserines SYNGENTA PARTICIPATIONS AG (CH) 2017-05-09 US disclosed
EP-3137449-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED CYCLOSERINES Syngenta Participations AG (CH) 2017-03-08 EP disclosed
US-20170044116-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED CYCLOSERINES SYNGENTA PARTICIPATIONS AG (CH) 2017-02-16 US disclosed
WO-2015166094-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED CYCLOSERINES SYNGENTA PARTICIPATIONS AG (CH) 2015-11-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170044116-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED CYCLOSERINES C1S, C1R, C5 CYP2D6 407/4885LMNA 2991/4885BLM 4430/4885
US-20170204072-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED CYCLOSERINES C1S, C1R, C5 CYP2D6 332/4885LMNA 2889/4885BLM 4345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.