SCHEMBL17226239

SCHEMBL17226239

Cc1ccc(NC(=O)c2cccc(C(F)(F)F)c2)cc1Oc1ccc2nc(NC(=O)C3=COC=CC=C3)sc2n1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
KDR P35968 4/20 0.44
TEK Q02763 2/20 0.44
BRAF P15056 11/20 0.42
CSF1R P07333 5/20 0.41
KIT P10721 3/20 0.40
PDGFRB P09619 1/20 0.40
DDR1 Q08345 1/20 0.40
LCK P06239 4/20 0.40
MAPK14 Q16539 4/20 0.40
JAK3 P52333 2/20 0.40
ABL1 P00519 1/20 0.40
SRC P12931 1/20 0.40
RAF1 P04049 2/20 0.40
BTK Q06187 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857561 0.84 BRAF (0.48) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL2858679 0.83 KDR (0.48) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL2855913 0.83 BTK (0.50) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL2855661 0.83 KDR (0.53) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL2858206 0.81 KDR (0.51) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL13185061 0.79 KDR (0.44) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL2859286 0.78 WNT3A (0.47) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL13184980 0.76 LCK (0.45) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL13184976 0.76 KDR (0.40) ALDH1A1KDRTEKBRAFCSF1R
SCHEMBL2857374 0.76 BRAF (0.53) KDRBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2184285-B1 HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2015-11-04 EP disclosed