SCHEMBL17233282

SCHEMBL17233282

COc1ccccc1/C=C/C(=O)c1cccnc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 1.00
CYP1A1 P04798 8/20 1.00
CYP1B1 Q16678 8/20 1.00
CYP2D6 P10635 7/20 1.00
CYP3A4 P08684 6/20 1.00
CAPN1 P07384 1/20 0.85
CTSL P07711 1/20 0.85
CTSB P07858 1/20 0.85
MAPT P10636 4/20 0.72
LMNA P02545 3/20 0.72
NPC1 O15118 3/20 0.72
RAB9A P51151 2/20 0.72
BCHE P06276 1/20 0.72
HPGD P15428 2/20 0.65
ALDH1A1 P00352 1/20 0.65
KMT2A Q03164 1/20 0.65
MAOB P27338 2/20 0.63
NR1H4 Q96RI1 1/20 0.62
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17233278 0.88 CYP1A1 (0.82) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL12306208 0.85 CYP1A1 (0.73) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL17232029 0.85 CYP1A2 (1.00) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL1723179 0.84 MAPT (1.00) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL1723180 0.84 MAPT (1.00) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL17233276 0.83 CYP1A1 (1.00) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL9567804 0.82 MAPT (0.70) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL3600036 0.81 CYP1A1 (0.67) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL3600030 0.81 CYP1A1 (0.67) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4
SCHEMBL3597959 0.80 MAPT (0.72) CYP1A2CYP1A1CYP1B1CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015166043-A1 COMPOUNDS DE MONTFORT UNIVERSITY (GB) 2015-11-05 WO disclosed