SCHEMBL1723735

SCHEMBL1723735

CC(C)(C(=O)O)C(=O)Cc1ccc(-c2cnc(Nc3cccc(F)c3)nc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.45
SYK P43405 4/20 0.45
BTK Q06187 2/20 0.42
BLK P51451 1/20 0.42
SRC P12931 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
WNT3A P56704 3/20 0.41
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CCND2 P30279 1/20 0.40
CCND3 P30281 1/20 0.40
CDC7 O00311 2/20 0.40
LCK P06239 1/20 0.40
DAPK3 O43293 1/20 0.40
PRKD3 O94806 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL180770 0.80 HDAC3 (0.46) CNR2SYKBTKHDAC3HDAC1
SCHEMBL29818135 0.70 NPC1 (0.63) BTKBLKSRCHDAC3HDAC1
SCHEMBL180787 0.69 DGAT1 (0.64)
SCHEMBL16546762 0.69 DGAT1 (0.64)
SCHEMBL13664059 0.69 DGAT1 (0.64)
SCHEMBL1736682 0.68 GFRA3 (0.54) CNR2SYKHDAC3HDAC1HDAC2
SCHEMBL180650 0.67 DGAT1 (0.69) TBK1
SCHEMBL1448287 0.67 DGAT1 (0.50) SYKHDAC3HDAC1HDAC2HDAC6
SCHEMBL5459434 0.67 MEN1 (0.52) SYKSRCTP53PDE4BPDE4D
SCHEMBL1734253 0.67 CSNK2A1 (0.54) SYKHDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2404905-A1 New compounds Novartis AG (CH) 2012-01-11 EP disclosed