SCHEMBL1723896

SCHEMBL1723896

CC(=O)C1CN(Cc2ccccc2)CC1c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.58
SLC6A4 P31645 1/20 0.47
S1PR5 Q9H228 2/20 0.47
S1PR1 P21453 1/20 0.47
MC4R P32245 3/20 0.46
ACHE P22303 1/20 0.45
ALDH1A1 P00352 1/20 0.45
SLC6A12 P48065 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
MCHR1 Q99705 1/20 0.44
SIGMAR1 Q99720 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1713398 1.00 RORC (0.58) RORCSLC6A4S1PR5S1PR1MC4R
SCHEMBL7997778 0.91 RORC (0.61) RORCS1PR5S1PR1SIGMAR1
SCHEMBL7832811 0.91 RORC (0.61) RORCS1PR5S1PR1SIGMAR1
SCHEMBL7883236 0.91 RORC (0.61) RORCS1PR5S1PR1SIGMAR1
SCHEMBL23923989 0.90 RORC (0.60) RORCSLC6A4S1PR5S1PR1SLC6A12
SCHEMBL15397505 0.90 RORC (0.60) RORCSLC6A4S1PR5S1PR1SLC6A12
SCHEMBL15397506 0.90 RORC (0.60) RORCSLC6A4S1PR5S1PR1SLC6A12
SCHEMBL1344658 0.88 RORC (0.59) RORCS1PR5S1PR1MC4R
SCHEMBL1443765 0.88 RORC (0.59) RORCS1PR5S1PR1MC4R
SCHEMBL3346208 0.87 RORC (0.58) RORCSLC6A4S1PR5MC4RSLC6A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185540-B1 PYRROLIDINE ARYL-ETHER AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-07-20 EP disclosed