SCHEMBL17241997

SCHEMBL17241997

NC(=O)c1cccnc1Oc1ccc(N)cc1

nearest known ligand 0.76

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.76
ALDH1A1 P00352 2/20 0.55
TDP1 Q9NUW8 1/20 0.52
ROCK2 O75116 6/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
APAF1 O14727 1/20 0.50
KMT2A Q03164 1/20 0.50
PARP10 Q53GL7 1/20 0.49
DRD1 P21728 1/20 0.48
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL742272 0.87 RAB9A (0.75) RAB9AALDH1A1TDP1ROCK2KDM4E
SCHEMBL6455377 0.86 RAB9A (0.74) RAB9AALDH1A1TDP1ROCK2KDM4E
SCHEMBL4165132 0.86 RAB9A (0.74) RAB9AALDH1A1TDP1ROCK2KDM4E
SCHEMBL28662140 0.86 RAB9A (1.00) RAB9AALDH1A1TDP1ROCK2KDM4E
Hydrochloric Acid SCHEMBL6831509 0.86 RAB9A (0.73) RAB9AALDH1A1TDP1ROCK2KDM4E
SCHEMBL6120093 0.85 RAB9A (0.72) RAB9AALDH1A1TDP1ROCK2KDM4E
SCHEMBL3692391 0.84 RAB9A (0.67) RAB9AALDH1A1ROCK2KDM4E
SCHEMBL30678410 0.84 RAB9A (0.70) RAB9AALDH1A1TDP1ROCK2KDM4E
SCHEMBL3699763 0.84 RAB9A (0.70) RAB9AALDH1A1TDP1ROCK2KDM4E
SCHEMBL620646 0.84 TDP1 (0.76) RAB9AALDH1A1TDP1MEN1APAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085482-B Substituted diethylenediamine compound and its application method and purposes 广东东阳光药业有限公司 2018-08-10 CN disclosed
WO-2015169180-A1 SUBSTITUTED PIPERAZINE COMPOUNDS AND METHODS AND USE THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2015-11-12 WO disclosed