SCHEMBL17255449

SCHEMBL17255449

COc1ccc(CNc2cncc(C(C)(C)C)n2)c(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 15/20 0.53
CYP3A4 P08684 15/20 0.53
CYP2D6 P10635 14/20 0.53
CYP2C19 P33261 14/20 0.53
TSHR P16473 13/20 0.53
CLK4 Q9HAZ1 8/20 0.53
LMNA P02545 7/20 0.53
USP2 O75604 6/20 0.53
HSD17B10 Q99714 5/20 0.53
ALOX15 P16050 4/20 0.53
APLNR P35414 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
MAPK1 P28482 6/20 0.48
CYP2C9 P11712 4/20 0.48
ALDH1A1 P00352 5/20 0.48
KDM4C Q9H3R0 1/20 0.48
CASP7 P55210 1/20 0.47
GLA P06280 1/20 0.47
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17441855 0.82 CYP1A2 (0.55) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL2720254 0.79 CYP1A2 (0.52) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL15884679 0.77 APLNR (0.50) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL20238802 0.76 CYP1A2 (0.63) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL558073 0.76 FGFR3 (0.56) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL558386 0.76 PDGFRB (0.54) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL558361 0.75 CYP1A2 (0.53) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL558094 0.75 CYP1A2 (0.53) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL20092723 0.74 CYP1A2 (0.55) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL16368537 0.73 CYP1A2 (0.62) CYP1A2CYP3A4CYP2D6CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2944637-B1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM CORP (JP) 2020-02-19 EP disclosed
EP-2944637-A1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM Corporation (JP) 2015-11-18 EP disclosed
CN-104903320-A Nitrogen-containing heterocylic compound or salt thereof FUJIFILM CORP 2015-09-09 CN disclosed