SCHEMBL17259265

SCHEMBL17259265

CCc1c(CNS(=O)(=O)c2ccccc2)nn(-c2ccccc2)c1CC(C)C

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 5/20 0.76
KCNH2 Q12809 5/20 0.58
CACNA1G O43497 4/20 0.58
HTR6 P50406 7/20 0.49
KEAP1 Q14145 1/20 0.39
GLA P06280 1/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17259229 0.86 CACNA1H (1.00) CACNA1HKCNH2CACNA1GHTR6KEAP1
SCHEMBL17259271 0.81 CACNA1H (0.49) CACNA1HKCNH2CACNA1GHTR6KMT2A
SCHEMBL17259280 0.77 CACNA1H (0.46) CACNA1HKCNH2CACNA1GKMT2A
SCHEMBL17259219 0.76 CACNA1H (0.79) CACNA1HKCNH2CACNA1GHTR6KMT2A
SCHEMBL17259260 0.74 KCNH2 (1.00) CACNA1HKCNH2CACNA1GHTR6
SCHEMBL23400209 0.72 CACNA1H (0.43) CACNA1HKCNH2CACNA1GPOLB
SCHEMBL17259283 0.71 KDM4C (0.46) CACNA1HKCNH2CACNA1GHTR6POLB
SCHEMBL23401081 0.69 CACNA1H (0.48) CACNA1HKCNH2CACNA1GPOLB
SCHEMBL11249623 0.69 CACNA1H (0.48) CACNA1HKCNH2CACNA1GPOLB
SCHEMBL17259246 0.68 KCNH2 (0.87) CACNA1HKCNH2CACNA1GHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9493423-B2 Compounds capable of inhibiting voltage gated calcium ion channel, and pharmaceutical compositions comprising the same KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2016-11-15 US claimed
US-20150329533-A1 COMPOUNDS CAPABLE OF INHIBITING VOLTAGE GATED CALCIUM ION CHANNEL, AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2015-11-19 US claimed
US-9493423-B2 Compounds capable of inhibiting voltage gated calcium ion channel, and pharmaceutical compositions comprising the same KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2016-11-15 US disclosed
US-20150329533-A1 COMPOUNDS CAPABLE OF INHIBITING VOLTAGE GATED CALCIUM ION CHANNEL, AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2015-11-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150329533-A1 COMPOUNDS CAPABLE OF INHIBITING VOLTAGE GATED CALCIUM ION CHANNEL, AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CACNA1B, CACNA1F, CACNA1G CACNA1H 9/4885KCNH2 33/4885CACNA1G 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.