SCHEMBL1727033

SCHEMBL1727033

CCOC(=O)c1cc2[nH]c(Nc3cc(CNC(=O)C4(C(F)(F)F)CC4)ccc3Cl)nc2cc1OCC(F)F

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGES O14684 17/20 0.56
P2RY12 Q9H244 1/20 0.37
PDE5A O76074 2/20 0.33
PDE6D O43924 1/20 0.33
PDE6A P16499 1/20 0.33
PDE6G P18545 1/20 0.33
PDE6B P35913 1/20 0.33
PDE6C P51160 1/20 0.33
PDE6H Q13956 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3099526 0.97 PTGES (0.58) PTGESP2RY12
SCHEMBL11962197 0.90 PTGES (0.49) PTGESP2RY12
SCHEMBL3101702 0.85 PTGES (0.73) PTGES
SCHEMBL3100739 0.84 PTGES (0.79) PTGES
SCHEMBL3099096 0.83 PTGES (0.58) PTGES
SCHEMBL11961902 0.80 PTGES (0.63) PTGES
SCHEMBL15379477 0.76 PTGES (0.61) PTGES
SCHEMBL9939820 0.74 PTGES (0.44) PTGES
SCHEMBL9939985 0.74 PTGES (0.45) PTGES
SCHEMBL3106287 0.74 PTGES (0.47) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403852-A1 3H-IMIDAZO [4, 5 -C]PYRIDINE- 6 -CARBOXAMIDES AS ANTI- INFLAMMATORY AGENTS Boehringer Ingelheim International GmbH (DE) 2012-01-11 EP disclosed
WO-2010100249-A1 3H-IMIDAZO [4, 5 -C] PYRIDINE- 6 -CARBOXAMIDES AS ANTI- INFLAMMATORY AGENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-10 WO disclosed