SCHEMBL17277553

SCHEMBL17277553

CCc1cc(OC(F)(F)F)cc(S(=O)(=O)NCCN)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
FFAR4 Q5NUL3 2/20 0.39
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
MMP14 P50281 2/20 0.36
ADAM17 P78536 2/20 0.36
MMP1 P03956 1/20 0.36
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
SLC6A2 P23975 1/20 0.34
KAT6A Q92794 1/20 0.34
NAMPT P43490 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17277617 0.85 FFAR4 (0.48) CYP3A4L3MBTL1FFAR4BCHEACHE
SCHEMBL12062342 0.83 CYP3A4 (0.39) CYP3A4L3MBTL1FFAR4SLC6A4SLC6A3
SCHEMBL12075868 0.81 CYP3A4 (0.42) CYP3A4L3MBTL1FFAR4CA12CA1
SCHEMBL17277532 0.77 TP53 (0.36) CYP3A4FFAR4BCHEACHESLC6A4
SCHEMBL12075807 0.73 SCN8A (0.41) L3MBTL1
SCHEMBL12075491 0.72 KMT2A (0.53) CYP3A4
SCHEMBL17365350 0.71 BCHE (0.32) CYP3A4FFAR4BCHEACHESLC6A4
SCHEMBL21190211 0.71 TSHR (0.41) L3MBTL1SLC6A4
SCHEMBL3684870 0.70 CA12 (0.58) L3MBTL1FFAR4MMP2MMP9MMP14
SCHEMBL17277356 0.68 SLC7A5 (0.35) CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9193731-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2015-11-24 US disclosed