SCHEMBL12075868

SCHEMBL12075868

CCc1cc(C(F)(F)F)cc(S(=O)(=O)NCCN)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
CYP19A1 P11511 1/20 0.39
CYP2D6 P10635 1/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
GPBAR1 Q8TDU6 3/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
PPARG P37231 1/20 0.36
ERBB2 P04626 3/20 0.36
ERBB4 Q15303 3/20 0.36
FFAR4 Q5NUL3 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17277472 0.83 CYP3A4 (0.44) CYP3A4CYP19A1CYP2D6PSEN1PSEN2
SCHEMBL12062350 0.83 CYP3A4 (0.44) CYP3A4CYP19A1CYP2D6PSEN1PSEN2
SCHEMBL17277553 0.81 CYP3A4 (0.40) CYP3A4CA1CA2FFAR4L3MBTL1
SCHEMBL12075491 0.77 KMT2A (0.53) CYP3A4CYP19A1ALDH1A1
SCHEMBL24454595 0.74 LMNA (0.38) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL17115760 0.74 CYP3A4 (0.64) CYP3A4CYP19A1CA1CA2ALDH1A1
SCHEMBL13753684 0.74 MEN1 (0.50) CYP3A4CYP19A1CYP2D6PSEN1PSEN2
SCHEMBL30230186 0.72 PSEN1 (0.48) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL12062342 0.72 CYP3A4 (0.39) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL1788802 0.71 SMN1; SMN2 (0.40) CYP3A4CYP19A1CYP2D6PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9193731-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2015-11-24 US disclosed
US-20120220566-A1 Antimicrobial Compounds and Methods of Making and Using the Same RIB-X PHARMACEUTICALS, INC. (US) 2012-08-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120220566-A1 Antimicrobial Compounds and Methods of Making and Using the Same MPO, LPO, CAT CYP3A4 1470/4885CYP19A1 2570/4885CYP2D6 993/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.