SCHEMBL17286240

SCHEMBL17286240

CCCCNc1nc(N)nnc1Cl

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 19/20 0.62
TLR7 Q9NYK1 11/20 0.62
KDM4E B2RXH2 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17286238 0.82 KDM4E (0.54) TLR8TLR7KDM4ENPSR1L3MBTL1
SCHEMBL18286678 0.81 TLR8 (0.65) TLR8TLR7
SCHEMBL8695685 0.79 TLR8 (0.64) TLR8TLR7L3MBTL1
SCHEMBL11752787 0.79 TLR8 (0.73) TLR8TLR7L3MBTL1
SCHEMBL19495041 0.78 TLR8 (0.71) TLR8TLR7
SCHEMBL17286218 0.77 TLR8 (1.00) TLR8TLR7
SCHEMBL20434302 0.77 TLR8 (0.69) TLR8TLR7L3MBTL1
SCHEMBL17035544 0.76 TLR8 (0.59) TLR8TLR7L3MBTL1
SCHEMBL20434277 0.75 TLR8 (1.00) TLR8TLR7
SCHEMBL17693700 0.74 TLR8 (0.57) TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903976-B1 1,2,4-TRIAZINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS. CENTRE NAT DE LA RECH SCIENT (C N R S ) (FR) 2016-12-07 EP disclosed
US-9416114-B2 1,2,4-triazine derivatives for the treatment of viral infections CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2016-08-16 US disclosed
US-20150336907-A1 1,2,4-TRIAZINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS UNIVERSITE DE ROUEN (FR) 2015-11-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150336907-A1 1,2,4-TRIAZINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS MAVS, IL5, ZC3HAV1 TLR8 177/4885TLR7 51/4885KDM4E 1588/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.