Bromide

Bromide

SCHEMBL1731813

Br.CCCN1CCOc2c1cc(C(=O)CN1Cc3ccc(CC)nc3C1=N)cc2C(C)(C)C

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
F2R P25116 13/20 0.40
PTGS2 P35354 4/20 0.33
PTGS1 P23219 3/20 0.33
ALOX5 P09917 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL1730761 0.94 F2R (0.41) F2RPTGS2PTGS1ALOX5
Bromide SCHEMBL5488877 0.93 F2R (0.39) F2RPTGS2PTGS1ALOX5
Bromide SCHEMBL1730915 0.92 F2R (0.40) F2RPTGS2PTGS1ALOX5
Bromide SCHEMBL5485459 0.92 F2R (0.38) F2RPTGS2PTGS1ALOX5
Hydrochloric Acid SCHEMBL5488919 0.92 F2R (0.38) F2RPTGS2PTGS1ALOX5
Bromide SCHEMBL1729538 0.88 F2R (0.39) F2RPTGS2PTGS1ALOX5
Bromide SCHEMBL1730039 0.86 F2R (0.37) F2R
Bromide SCHEMBL1732301 0.85 PTGS2 (0.45) F2RPTGS2PTGS1ALOX5
Bromide SCHEMBL1731907 0.85 F2R (0.36) F2RPTGS2PTGS1ALOX5
Bromide SCHEMBL1731616 0.83 PTGS2 (0.47) F2RPTGS2PTGS1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1391451-B1 2-IMINOPYRROLIDINE DERIVATES EISAI R&D MAN CO LTD (JP) 2011-11-23 EP disclosed